Cemiplimab

Cemiplimab
Monoclonal antibody
TypeWhole antibody
SourceHuman
TargetPD-1
Clinical data
Pronunciationsem' ip li" mab
Trade namesLibtayo
Other namesREGN-2810, REGN2810, cemiplimab-rwlc
AHFS/Drugs.comMonograph
MedlinePlusa618054
License data
Pregnancy
category
  • AU: D
Routes of
administration
Intravenous
ATC code
Legal status
Legal status
  • AU: S4 (Prescription only)
  • CA: ℞-only / Schedule D
  • US: ℞-only
  • EU: Rx-only
  • In general: ℞ (Prescription only)
Pharmacokinetic data
Elimination half-life19 days
Identifiers
CAS Number
DrugBank
ChemSpider
  • none
UNII
KEGG
Chemical and physical data
FormulaC6380H9808N1688O2000S44
Molar mass143569.10 g·mol−1

Cemiplimab, sold under the brand name Libtayo, is a monoclonal antibody medication used for the treatment of squamous cell skin cancer. Cemiplimab belongs to a class of drugs that binds to the programmed death receptor-1 (PD-1), blocking the PD-1/PD-L1 pathway.

The most common side effects include fatigue, rash, diarrhea, musculoskeletal pain, and nausea.

It was approved for medical use in the United States in September 2018, in the European Union in June 2019. and in Australia in July 2020.

Cemiplimab is the first approval by the US Food and Drug Administration of a medication specifically for advanced cutaneous squamous cell carcinoma. Cemiplimab is a therapeutic alternative on the World Health Organization's List of Essential Medicines.